2016年9月5日星期一
U-47700(Power)
U-47700 is an opioid analgesic drug developed by a team at Upjohn in the 1970s. U-47700 was derived from an earlier opioid AH-7921. U-47700 is selective for the µ-opioid receptor with a Kd value of 5.3 nM compared to 910 nM for the κ-opioid receptor and has around 7.5 x the potency of morphine in animal models.
1 | Product name | U-47700 | |
2 | Full chemical name | trans-3,4-dichloro-N-(2-(dimethylamino)cyclohexyl)-N-methylbenzamide | |
3 | Formal Name | ||
4 | CAS num | 121348-98-9 | |
5 | Molecular Formula |
| |
6 | Average mass | 329.265 g/mol | |
7 | Purity | ≥99.1% | |
8 | Stability | 2 years | |
9 | Storage | -20°C | |
10 | Formulation A powder solid | ||
11 | λmax 221, 315 nm | ||
12 | Shipping Wet ice in continental US; may vary elsewhere |
my contact information is:
Email: cloris_2016@tuskwei.com
Skype: betty_3451
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Acrylfentanyl
Acrylfentanyl (also known as acryloylfentanyl) is a highly potent opioid analgesic that is an analog of fentanyland has been sold online as a designer drug. In animal studies the IC50 or half maximal inhibitory concentration for acrylfentanyl to displace naloxone is 1.4 nM, being slightly more potent than fentanyl itself (1.6 nM) as well as having a longer duration of action.
TECHNICAL INFORMATION
Formal Name | N-phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]-2-propenamide, monohydrochloride |
CAS Number | 79279-03-1 |
Molecular Formula | C22H26N2O • HCl |
Formula Weight | 370.9 |
Purity | ≥98% |
Formulation | A neat solid |
SMILES | O=C(N(C1=CC=CC=C1)C2CCN(CCC3=CC=CC=C3)CC2)C=C.Cl |
InChI Code | 1S/C22H26N2O.ClH/c1-2-22(25)24(20-11-7-4-8-12-20)21-14-17-23(18-15-21)16-13-19-9-5-3-6-10-19;/h2-12,21H,1,13-18H2;1H |
InChI Key | YUHNRLIKLNYPDD-UHFFFAOYSA-N |
WARNING - This product is not for human or veterinary use.
SHIPPING & STORAGE
Storage | -20°C |
Shipping | Room temperature in continental US; may vary elsewhere |
Stability | As supplied, 3 years from the QC date provided on the Certificate of Analysis, when stored properly |
my contact information is:
Email: cloris_2016@tuskwei.com
Skype: betty_3451
website is: http://www.tuskwei.cn/content.asp?id=51
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