显示标签为“opioid analgesic”的博文。显示所有博文
显示标签为“opioid analgesic”的博文。显示所有博文

2016年9月5日星期一

Furanylfentanyl (Fu-F)






Furanylfentanyl (Fu-F) is an opioid analgesic which has an ED50 value of 0.02mg/kg in mice.

Appearance: White powder

Purity: >99%

Package: 1kg/Aluminum foil bag or as customer's request.

Application: For chemical research

Production Capacity: 500 Kilogram/Month

Storage: Kept in a cool,dry and ventilated place

Side effects of fentanyl analogs are similar to those of fentanyl itself, which include itching, nausea and potentially serious respiratory depression, which can be life-threatening. Fentanyl analogs have killed hundreds of people throughout Europe and the former Soviet republics since the most recent resurgence in use began in Estonia in the early 2000s, and novel derivatives continue to appear.

Life-threatening adverse reactions due to furanylfentanyl use have been observed in Sweden. At least seven deaths in Cook County, Illinois, have been linked to furanylfentanyl.

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U-47700(Power)





U-47700 is an opioid analgesic drug developed by a team at Upjohn in the 1970s. U-47700 was derived from an earlier opioid AH-7921. U-47700 is selective for the µ-opioid receptor with a Kd value of 5.3 nM compared to 910 nM for the κ-opioid receptor and has around 7.5 x the potency of morphine in animal models.
1Product nameU-47700
2Full chemical nametrans-3,4-dichloro-N-(2-(dimethylamino)cyclohexyl)-N-methylbenzamide
3Formal Name 
4CAS num121348-98-9
5Molecular Formula
C16H22Cl2N2O
6 Average mass329.265 g/mol
7Purity ≥99.1%
8Stability 2 years
9Storage -20°C
10Formulation A powder solid
11λmax 221, 315 nm
12Shipping Wet ice in continental US; may vary elsewhere

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Acrylfentanyl


Acrylfentanyl (also known as acryloylfentanyl) is a highly potent opioid analgesic that is an analog of fentanyland has been sold online as a designer drug. In animal studies the IC50 or half maximal inhibitory concentration for acrylfentanyl to displace naloxone is 1.4 nM, being slightly more potent than fentanyl itself (1.6 nM) as well as having a longer duration of action.
TECHNICAL INFORMATION
Formal NameN-phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]-2-propenamide, monohydrochloride
CAS Number79279-03-1
Molecular FormulaC22H26N2O • HCl
Formula Weight370.9
Purity≥98%
FormulationA neat solid
SMILESO=C(N(C1=CC=CC=C1)C2CCN(CCC3=CC=CC=C3)CC2)C=C.Cl
InChI Code1S/C22H26N2O.ClH/c1-2-22(25)24(20-11-7-4-8-12-20)21-14-17-23(18-15-21)16-13-19-9-5-3-6-10-19;/h2-12,21H,1,13-18H2;1H
InChI KeyYUHNRLIKLNYPDD-UHFFFAOYSA-N
WARNING - This product is not for human or veterinary use.
SHIPPING & STORAGE
Storage-20°C
ShippingRoom temperature in continental US; may vary elsewhere
StabilityAs supplied, 3 years from the QC date provided on the Certificate of Analysis, when stored properly

my contact information is: 

Email: cloris_2016@tuskwei.com 

Skype: betty_3451

website is: http://www.tuskwei.cn/content.asp?id=51